PD 145065
A highly potent but non-selective endothelin receptor antagonist [IC50 = 4 nM for the ETA receptor (rabbit renal artery vascular smooth muscle cells); IC50 = 15 nM for the ETB receptor (rat cerebellum)].
產(chǎn)品信息
Peptide Sequence  Ac-D-Bhg-Leu-Asp-Ile-Ile-Trp-OH (Bhg = 5H-dibenzo[a,d]cycloheptene-5-glycine)
Form  White solid
Molar mass  992.1
Purity  ≥98% by HPLC
Solubility  Phosphate Buffer, pH 7.5
Chemical formula  C52H63N7O10 · 2Na
CAS number  153049-49-1
商店和運輸信息
Storage  +2°C to +8°C
Ship  Ambient Temperature Only
Standard Handling