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WNT SYNERGIST, QS11

產(chǎn)品編號(hào): 681668-5MG     查看說明書
產(chǎn)品名稱: WNT SYNERGIST, QS11  .0   訂購此產(chǎn)品 
供應(yīng)商: Merck
規(guī)格: ***
目錄價(jià): 4551
庫存狀態(tài): 3周到貨
CAS編號(hào): 944328-88-5
應(yīng)用范圍: 生化實(shí)驗(yàn)
種屬來源:
相關(guān)信息:

Wnt Synergist, QS11
QS11, Wnt Pathway Activator II
A cell-permeable purine compound that binds ARFGAPs (Kd = 364 and 620 nM for AMAP1 and ARFGAP1, respectively) and acts as a broad specificity ARFGAPs inhibitor (GTPase activating proteins of ADP-ribosylation factor). Shown to synergize with Wnt-3a and specifically activate the canonical Wnt/β-catenin signaling pathway both in vitro (2-, 40-, and 200-fold increase of basal transcription activity by QS11, Wnt-3a, and QS11/Wnt-3a, respectively, in a Super(8X)TOPFlash reporter assay using HEK293 cells) and in vivo (in the induction of Xenopus embryonic axis duplication). Also reported to block the migration of AMAP1-overexpressing MDA-MB-231 cells (86% inhibition at 2.5 µM).
產(chǎn)品信息
Form  Pale amber solid
Molar mass  567.7
Protect from Light  是的
Packaged under inert gas  是的
Purity  ≥95% by HPLC
Solubility  DMSO or EtOH
Chemical formula  C36H33N5O2
CAS number  944328-88-5
商店和運(yùn)輸信息
Storage  +2°C to +8°C
Ship  Ambient Temperature Only
Regulatory Review

保存條件: 2°C - 8°C
說明書地址: 點(diǎn)擊查看詳細(xì)
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